A-61603 is a selective alpha1A/alpha1a-adrenergic receptor agonist with Ki of 8.89 nM for rat submaxillary gland alpha1A, Ki of 30.5 nM for cloned bovine alpha1a. A-61603 potentiates Ca2+ transients with EC50 of 6.9 nM. A-61603 stimulates phosphoinositide hydrolysis, induces contractile responses in vas deferens, prostate strips, and spleen strips, and exhibits low activity in aortic rings. A-61603 can be used for research on adrenergic function[1][2].
Molecular Weight:
390.30
Purity:
99.34
CAS Number:
[107756-30-9]
Formula:
C14H20BrN3O3S
Target:
Adrenergic Receptor
Application Notes:
MCE Product type: Reference compound
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