A-61603 is a selective alpha1A/alpha1a-adrenergic receptor agonist with Ki of 8.89 nM for rat submaxillary gland alpha1A, Ki of 30.5 nM for cloned bovine alpha1a. A-61603 potentiates Ca2+ transients with EC50 of 6.9 nM. A-61603 stimulates phosphoinositide hydrolysis, induces contractile responses in vas deferens, prostate strips, and spleen strips, and exhibits low activity in aortic rings. A-61603 can be used for research on adrenergic function[1][2].
Molekulargewicht:
390.30
Reinheit:
99.34
CAS Nummer:
[107756-30-9]
Formel:
C14H20BrN3O3S
Target-Kategorie:
Adrenergic Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten
