Compound 114 is a dual D3 dopamine and mu-opioid receptor antagonist with K i values of 46.5 nM and 691 nM, respectively. Its MOR partial agonism provides analgesic potential, while D3R antagonism may mitigate abuse liability, supporting research in neuropharmacology and addiction studies.
Molecular Weight:
420.38
Formula:
C22H27Cl2N3O
Target:
Dopamine Receptor,Opioid Receptor
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