Compound 121 is a dual D3 receptor antagonist (K i = 361 nM) and mu-opioid receptor antagonist/partial agonist (K i = 85.2 nM). This profile suggests utility in preclinical research for investigating novel analgesic mechanisms with potentially reduced abuse liability, applicable in both in vitro binding assays and in vivo behavioral models.
Molecular Weight:
410.98
Formula:
C25H31ClN2O
Target:
Dopamine Receptor,Opioid Receptor
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