EZH2-IN-14 is a selective inhibitor of EZH2 (histone methyltransferase) with an IC50 value of 12 nM. EZH2-IN-14 targets the histone methyltransferase EZH2, inhibiting its trimethylation of histone H3K27. In vitro, EZH2-IN-14 regulates gene expression in cancer cells, inhibits proliferation, and induces apoptosis, making it suitable for studying tumor epigenetic regulatory mechanisms and for potential drug development.
Molecular Weight:
541.69
Purity:
99.82%
CAS Number:
[1979157-17-9]
Formula:
C31H39N7O2
Target:
Histone Methyltransferase
T73134
T73134
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