Jaspamycin is a potent PKA activator that binds to the PKAR site of Trypanosoma brucei, with EC50 and Kd values of 6.5 nM and 8 nM, respectively. It does not bind to purified human PKARIalpha and shows favorable antiparasitic activity.
Molecular Weight:
292.25
CAS Number:
[22242-96-2]
Formula:
C12H12N4O5
Target:
PKA|||Parasite
T11711
T11711
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