Autophagy, LG 100064, LG100064, LG-100064, Inhibitor, inhibit, RAR/RXR, Retinoid X receptors, RetinoidReceptor, Retinoic acid receptors, Retinoid Receptor, RXRalpha, RXRbeta, RXRgamma
LG-100064 is a retinoid X receptor (RXR) agonist with EC50 values of 330 nM for RXRalpha, 200 nM for RXRbeta, and 260 nM for RXRgamma. It is used in research on nuclear receptor signaling, metabolic diseases, and cancer, facilitating in vitro transcriptional assays and in vivo studies in diabetes and atherosclerosis models.