PDHK1-IN-3 (Compound 29) is a selective inhibitor of PDHK1, demonstrating an IC50 of 0.028 µM for PDHK1 and an IC50 of 0.120 µM for PDHK2. It inhibits PDHK1 activity by forming a covalent bond with Lys299 in the enzyme. PDHK1-IN-3 is applicable to research on autoimmune diseases, inflammatory conditions, and cancer.
Target-Kategorie:
Dehydrogenase
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