ITI-214, CAS [[1642303-38-5]]
Artikelnummer:
BYT-ORB1309535
Produktübersicht
Artikelname:
ITI-214, CAS [[1642303-38-5]]
Artikelnummer:
BYT-ORB1309535
Hersteller Artikelnummer:
orb1309535
Alternativnummer:
BYT-ORB1309535-1,BYT-ORB1309535-10,BYT-ORB1309535-100,BYT-ORB1309535-2,BYT-ORB1309535-25,BYT-ORB1309535-5,BYT-ORB1309535-50
Hersteller:
Biorbyt
Kategorie:
Biochemikalien
Alternative Synonym:
cognitive, CNS-active, PDE, PDE1, oral, inhibit, ITI214, ITI-214, ITI 214, motor, Inhibitor, selective, phosphodiesterase, Phosphodiesterase (PDE)
Produktbeschreibung
ITI-214 is a highly potent and selective picomolar inhibitor of PDE1 (Ki = 58 pM), demonstrating minimal off-target activity. This tool compound is valuable for investigating PDE1s role in neurological and cardiovascular research, with utility in both cellular assays and animal models.
Produkteigenschaften
Molekulargewicht:
605.56
Reinheit:
98.21% (May vary between batches)
CAS Nummer:
[1642303-38-5]
Formel:
C29H29FN7O5P
Target-Kategorie:
PDE
Anwendungsbeschreibung
Anwendungsbeschreibung:
Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (3.3 mM),DMSO:30 mg/mL (49.54 mM)