TAS4464 hydrochloride, CAS [[1848959-11-4]]

Artikelnummer: BYT-ORB1309030
Artikelname: TAS4464 hydrochloride, CAS [[1848959-11-4]]
Artikelnummer: BYT-ORB1309030
Hersteller Artikelnummer: orb1309030
Alternativnummer: BYT-ORB1309030-1,BYT-ORB1309030-10,BYT-ORB1309030-100,BYT-ORB1309030-25,BYT-ORB1309030-5,BYT-ORB1309030-50
Hersteller: Biorbyt
Kategorie: Biochemikalien
Alternative Synonym: Inhibitor, NEDD8-activating Enzyme, NEDD8, NAE, inhibit, E1Enzyme, E1 Enzyme, E2 Enzyme, E2Enzyme, E3 Enzyme, E3Enzyme, TAS4464, TAS-4464, TAS4464 Hydrochloride, TAS4464 hydrochloride, TAS-4464 Hydrochloride, TAS-4464 hydrochloride, TAS 4464, TAS 4464 Hydrochloride
TAS4464 hydrochloride is a potent and selective NEDD8-activating enzyme (NAE) inhibitor with an IC50 of 0.955 nM. It is a valuable research tool for investigating the neddylation pathway in oncology research, demonstrating activity in both cellular and in vivo models of cancer.
Molekulargewicht: 542.97
Reinheit: 98.96% (May vary between batches)
CAS Nummer: [1848959-11-4]
Formel: C21H24ClFN6O6S
Target-Kategorie: NEDD8,E1/E2/E3 Enzyme
Anwendungsbeschreibung: Solubility: 30% PEG300+70% Saline:5 mg/mL (9.21 mM),H2O:4 mg/mL (7.37 mM),DMSO:80 mg/mL (147.34 mM)